SCHEMBL17277752

SCHEMBL17277752

CC(=O)c1cc(Cl)c2cn[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.43
PRKAB2 O43741 1/20 0.41
PRKAG1 P54619 1/20 0.41
PRKAA2 P54646 1/20 0.41
PRKAA1 Q13131 1/20 0.41
PRKAG3 Q9UGI9 1/20 0.41
PRKAG2 Q9UGJ0 1/20 0.41
PRKAB1 Q9Y478 1/20 0.41
MAOB P27338 8/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
GRK2 P25098 1/20 0.37
IDO1 P14902 1/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
METAP2 P50579 1/20 0.36
JAK2 O60674 2/20 0.36
JAK1 P23458 2/20 0.36
TYK2 P29597 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1759083 0.85 TTR (0.46) NOS1MAOBALDH1A1IDO1METAP2
SCHEMBL13132270 0.83 TDO2 (0.50) NOS1MAOBKDM4EALDH1A1MAPT
SCHEMBL12664045 0.83 NOS1 (0.40) NOS1MAOBGRK2IDO1METAP2
SCHEMBL12647460 0.83 NOS1 (0.40) NOS1MAOBGRK2IDO1JAK2
SCHEMBL4410091 0.78 LMNA (0.50) MAOBKDM4EALDH1A1MAPTMETAP2
SCHEMBL18508895 0.73 NOS1 (0.37) NOS1MAOBGRK2IDO1METAP2
SCHEMBL14487466 0.72 METAP2 (0.56) NOS1IDO1METAP2
SCHEMBL16618130 0.69 IDO1 (0.61) NOS1IDO1METAP2
SCHEMBL7572191 0.69 NOS1 (0.50) NOS1KDM4EALDH1A1MAPTIDO1
SCHEMBL31190826 0.69 METAP2 (0.53) NOS1IDO1METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2947082-A1 N1-PYRAZOLOSPIROKETONE ACETYL-CoA CARBOXYLASE INHIBITORS Pfizer Inc (US) 2015-11-25 EP disclosed