SCHEMBL4411259

SCHEMBL4411259

COc1ccc2c(COc3cccc4[nH]c(OC(=O)NC5CCN(C[C@@H]6CCCN7CCCC[C@H]67)CC5)cc34)coc2c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.40
ALDH1A1 P00352 5/20 0.36
MCHR1 Q99705 1/20 0.36
LTA4H P09960 3/20 0.35
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 3/20 0.33
CCR3 P51677 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CXCR3 P49682 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SIGMAR1 Q99720 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4410339 0.91 MAOB (0.34) MAOBALDH1A1MCHR1MEN1KMT2A
Hydrochloric Acid SCHEMBL4409030 0.91 ALDH1A1 (0.37) MAOBALDH1A1LTA4HSMN1; SMN2
Hydrochloric Acid SCHEMBL4397030 0.90 DRD2 (0.35) MAOBALDH1A1
Hydrochloric Acid SCHEMBL4406718 0.90 ALDH1A1 (0.32) MAOBALDH1A1LMNA
SCHEMBL13593470 0.90 MAOB (0.43) MAOBALDH1A1MCHR1LTA4HKMT2A
SCHEMBL4404574 0.90 ALDH1A1 (0.34) MAOBALDH1A1MCHR1KMT2A
SCHEMBL913973 0.90 MAOB (0.43) MAOBALDH1A1MCHR1LTA4HKMT2A
Hydrochloric Acid SCHEMBL4406706 0.89 ALDH1A1 (0.34) ALDH1A1MCHR1KMT2A
SCHEMBL4403829 0.88 MAOB (0.44) MAOBALDH1A1MCHR1LTA4HMEN1
SCHEMBL4396348 0.88 SOS1 (0.34) MAOBALDH1A1MCHR1SMN1; SMN2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed