SCHEMBL4403829

SCHEMBL4403829

COc1ccc2c(COc3cccc4[nH]c(OC(=O)NC5CCN(CCN6CCCCCC6)CC5)cc34)coc2c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.44
ALDH1A1 P00352 5/20 0.39
MCHR1 Q99705 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
LTA4H P09960 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAPT P10636 2/20 0.37
DRD2 P14416 1/20 0.37
DRD3 P35462 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4401840 0.94 MAOB (0.44) MAOBALDH1A1MCHR1LTA4HMEN1
SCHEMBL4396402 0.94 MAOB (0.44) MAOBALDH1A1MCHR1MEN1KMT2A
SCHEMBL4409300 0.89 MAOB (0.44) MAOBMCHR1DRD2DRD3ACHE
SCHEMBL915839 0.89 MAOB (0.47) MAOBALDH1A1MCHR1HRH3LTA4H
SCHEMBL4411259 0.88 MAOB (0.40) MAOBALDH1A1MCHR1LTA4HMEN1
SCHEMBL4406823 0.88 HTR4 (0.38) ALDH1A1MCHR1KMT2ADRD2DRD3
SCHEMBL4399337 0.86 MAOB (0.41) MAOBALDH1A1MCHR1LTA4HMAPT
SCHEMBL4396426 0.86 BDKRB1 (0.37) MAOBALDH1A1DRD2DRD3
SCHEMBL4400748 0.85 MAOB (0.37) MAOBALDH1A1MCHR1KMT2ADRD2
Hydrochloric Acid SCHEMBL4401842 0.84 MCHR1 (0.36) MCHR1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed