SCHEMBL4415503

SCHEMBL4415503

O=C1c2ccccc2C(=O)N1Cc1ccc(-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 4/20 0.65
ADRA1D P25100 2/20 0.60
ADRA1A P35348 2/20 0.60
ADRA1B P35368 2/20 0.60
CHRM3 P20309 1/20 0.57
CASP3 P42574 3/20 0.55
CA12 O43570 2/20 0.55
CA1 P00915 2/20 0.55
CA9 Q16790 2/20 0.55
HDAC1 Q13547 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CA2 P00918 1/20 0.51
MMP2 P08253 1/20 0.50
MMP9 P14780 1/20 0.50
HSP90AA1 P07900 1/20 0.49
PARK7 Q99497 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11167209 0.87 CASP3 (0.67) ADRA1DADRA1AADRA1BCASP3CA12
SCHEMBL1691386 0.83 CASP3 (0.68) ADRA1DADRA1AADRA1BCASP3CA12
SCHEMBL4424799 0.82 CASP3 (0.79) ADRA1DADRA1AADRA1BCASP3CA12
SCHEMBL31752583 0.81 KMT2A (0.56) CHRM5ADRA1DADRA1AADRA1BCHRM3
SCHEMBL19835813 0.81 CHRM5 (0.48) CHRM5ADRA1DADRA1AADRA1BCHRM3
SCHEMBL13448084 0.81 CA12 (0.58) CHRM5ADRA1DADRA1AADRA1BCASP3
SCHEMBL4424839 0.80 CES2 (0.61) ADRA1DADRA1AADRA1BCASP3CA12
SCHEMBL24827438 0.80 KMT2A (0.58) CHRM5ADRA1DADRA1AADRA1BCHRM3
SCHEMBL19925305 0.80 CASP3 (0.54) CHRM5ADRA1DADRA1AADRA1BCHRM3
SCHEMBL7957008 0.79 ADRA1D (0.62) CHRM5ADRA1DADRA1AADRA1BCHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479671-B1 Pyrimidinone compounds SMITHKLINE BEECHAM PLC (GB) 2009-05-27 EP disclosed
US-7115616-B2 Pyrimidinone compounds SMITHKLINE BEECHAM PLC (GB) 2006-10-03 US disclosed