SCHEMBL4415550

SCHEMBL4415550

CN(Cc1ccc(-c2ccc(Cl)cc2)cc1)C(=O)CBr

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.66
ALDH1A1 P00352 3/20 0.66
HTT P42858 2/20 0.66
AOC3 Q16853 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 3/20 0.45
MCHR1 Q99705 2/20 0.44
KDM4E B2RXH2 1/20 0.44
KMT2A Q03164 2/20 0.43
ERCC1 P07992 1/20 0.43
ERCC4 Q92889 1/20 0.43
MEN1 O00255 1/20 0.43
HTR2A P28223 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5867397 0.80 MTOR (0.49) RAB9AALDH1A1HTTAOC3NPC1
SCHEMBL9824635 0.80 ALDH1A1 (1.00) RAB9AALDH1A1HTTAOC3SMN1; SMN2
SCHEMBL3301637 0.78 NPC1 (0.72) RAB9AALDH1A1AOC3SMN1; SMN2NPC1
SCHEMBL9824160 0.77 ALDH1A1 (0.70) RAB9AALDH1A1HTTAOC3SMN1; SMN2
SCHEMBL6412640 0.75 ALDH1A1 (0.68) RAB9AALDH1A1HTTAOC3SMN1; SMN2
SCHEMBL11300231 0.74 ALDH1A1 (0.66) RAB9AALDH1A1HTTAOC3SMN1; SMN2
SCHEMBL8790300 0.73 CRHBP (0.51) RAB9AALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL296937 0.73 ALDH1A1 (0.64) RAB9AALDH1A1HTTSMN1; SMN2KMT2A
SCHEMBL10546564 0.73 ALDH1A1 (0.51) RAB9AALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL2056269 0.73 HRH3 (0.77) RAB9AALDH1A1HTTAOC3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479671-B1 Pyrimidinone compounds SMITHKLINE BEECHAM PLC (GB) 2009-05-27 EP disclosed
EP-1479671-A1 Pyrimidinone compounds SMITHKLINE BEECHAM PLC (GB) 2004-11-24 EP disclosed
EP-1175408-A1 PYRIMIDINONE COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 2002-01-30 EP disclosed
WO-2000066567-A1 PYRIMIDINONE COMPOUNDS SMITHKLINE BEECHAM PLC (GB) 2000-11-09 WO disclosed