SCHEMBL5867397

SCHEMBL5867397

CN(Cc1ccc(-c2ccc(C(F)(F)F)cc2)cc1)C(=O)CBr

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
LSS P48449 1/20 0.47
PTPN1 P18031 1/20 0.45
GSK3B P49841 1/20 0.45
TACR1 P25103 1/20 0.44
PYCR1 P32322 1/20 0.43
PPARA Q07869 1/20 0.43
RAB9A P51151 3/20 0.42
KIF11 P52732 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
NPC1 O15118 2/20 0.41
AOC3 Q16853 1/20 0.41
MAOB P27338 1/20 0.41
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4415550 0.80 RAB9A (0.66) MEN1KMT2ARAB9AALDH1A1HTT
SCHEMBL21789134 0.80 ALDH1A1 (0.66) MTORMEN1KMT2ALSSTACR1
SCHEMBL3880049 0.79 RAB9A (0.51) MTORMEN1KMT2ALSSTACR1
SCHEMBL7390057 0.76 MTOR (0.55) MTORMEN1KMT2ALSSTACR1
SCHEMBL2056267 0.76 HRH3 (0.68) LSSPYCR1KIF11ALDH1A1MAOB
SCHEMBL3301637 0.74 NPC1 (0.72) MEN1KMT2ARAB9AALDH1A1NPC1
SCHEMBL19013415 0.74 MTOR (0.63) MTORMEN1KMT2ALSSTACR1
SCHEMBL5643054 0.71 KMT2A (0.68) MTORMEN1KMT2ALSSRAB9A
SCHEMBL3885499 0.71 HPGD (0.50) MTORMEN1KMT2ALSSTACR1
SCHEMBL30435641 0.71 MTOR (0.59) MTORMEN1KMT2ALSSTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115616-B2 Pyrimidinone compounds SMITHKLINE BEECHAM PLC (GB) 2006-10-03 US disclosed
US-6953803-B1 1-[(N-(2-(diethylamino)ethyl)-N-(4-(4-trifluoromethylphenyl)benzyl)aminocarbonylmethyl)]-2-(4-fluorobenzyl)thio-5-(1-methyl-4-pyrazolylmethyl)pyrimidin-4-one; enzyme inhibitors of lipoprotein associated phospholipase A2 (Lp-PLA2); atherosclerosis SMITHKLINE BEECHAM P.L.C. (GB) 2005-10-11 US disclosed