SCHEMBL4418581

SCHEMBL4418581

CC(Cn1c(-c2c(F)cccc2F)c(Cl)nc(Cl)c1=O)S(C)(=O)=O

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 1/20 0.32
GNRHR P30968 12/20 0.32
MAPK14 Q16539 4/20 0.32
CYP3A4 P08684 1/20 0.32
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3986121 0.86 SMN1; SMN2 (0.39) ADORA2BGNRHRMAPK14
SCHEMBL4484784 0.76 SMN1; SMN2 (0.37) ADORA2BGNRHRMAPK14
SCHEMBL3913556 0.73 ALDH1A1 (0.40) GNRHR
SCHEMBL4493753 0.73 CASR (0.38) ADORA2BGNRHRMAPK14
SCHEMBL4478946 0.71 MAPT (0.43) CYP3A4
SCHEMBL3985349 0.71 ALDH1A1 (0.34) GNRHRMAPK14
SCHEMBL3986025 0.71 HCRTR1 (0.37) GNRHRMAPK14CYP3A4
SCHEMBL4483063 0.70 SYK (0.36) ADORA2BMAPK14
SCHEMBL3986451 0.70 JAK2 (0.36) ADORA2BGNRHRMAPK14
SCHEMBL4877540 0.70 TSHR (0.35) ADORA2BGNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2034993-A2 PYRAZINONES AS CELLULAR PROLIFERATION INHIBITORS E.I. DU PONT DE NEMOURS AND COMPANY (US) 2009-03-18 EP disclosed
WO-2007149448-A2 PYRAZINONES AS CELLULAR PROLIFERATION INHIBITORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2007-12-27 WO disclosed
EP-1848711-A1 FUNGICIDAL PYRAZINE DERIVATIVES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2007-10-31 EP disclosed
WO-2006089060-A1 FUNGICIDAL PYRAZINE DERIVATIVES E.I. DUPONT DE NEMOURS AND COMPANY (US) 2006-08-24 WO disclosed