SCHEMBL4426739

SCHEMBL4426739

CCCCC(C(=O)N[C@@H](CC(=O)O)c1ccccc1)n1cc(C)cc(Cc2cccc3ccccc23)c1=O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.42
CMA1 P23946 2/20 0.41
TACR3 P29371 2/20 0.38
IDH1 O75874 1/20 0.37
FPR1 P21462 5/20 0.35
FPR2 P25090 2/20 0.35
CTSA P10619 1/20 0.34
MAPT P10636 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGAV P06756 1/20 0.34
ITGA2B P08514 1/20 0.34
ITGB5 P18084 1/20 0.34
ITGB6 P18564 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4427172 0.93 CASP1 (0.43) CASP1CMA1TACR3IDH1FPR1
SCHEMBL4437254 0.90 FPR1 (0.36) CASP1CMA1FPR1FPR2CTSA
SCHEMBL4426944 0.88 FPR1 (0.39) CASP1FPR1FPR2CTSA
SCHEMBL4427187 0.88 MMP2 (0.38) CASP1FPR1CTSA
SCHEMBL7429087 0.88 MMP2 (0.38) CASP1FPR1CTSA
SCHEMBL4426794 0.88 CASP1 (0.39) CASP1TACR3FPR1CTSA
SCHEMBL6763118 0.85 CTSA (0.40) FPR1FPR2CTSA
SCHEMBL4435400 0.85 CTSA (0.40) FPR1CTSA
SCHEMBL8506622 0.85 CTSA (0.40) FPR1CTSA
SCHEMBL4435399 0.85 CTSA (0.40) FPR1CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1213288-B1 Propanoic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2009-01-14 EP disclosed