SCHEMBL4426765

SCHEMBL4426765

Fc1cccc(COc2cc(F)cc(F)c2)c1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOB P27338 14/20 0.67
NR4A2 P43354 2/20 0.59
MAOA P21397 2/20 0.59
IDO1 P14902 2/20 0.58
AGXT P21549 2/20 0.58
PARP10 Q53GL7 1/20 0.58
MRGPRX4 Q96LA9 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21944906 0.90 MAOB (0.59) MAOBNR4A2MAOAPARP10MRGPRX4
SCHEMBL11959694 0.85 MAOB (0.72) MAOBNR4A2MAOAIDO1AGXT
SCHEMBL27521276 0.85 MAOB (0.77) MAOBNR4A2MAOAIDO1AGXT
SCHEMBL18002578 0.84 MAOB (0.76) MAOBNR4A2MAOAPARP10
SCHEMBL24726478 0.84 MAOB (0.57) MAOBNR4A2MAOAPARP10MRGPRX4
SCHEMBL5042093 0.84 ALOX5 (0.55) MAOBMAOA
SCHEMBL12327547 0.84 MAOB (0.51) MAOBNR4A2MAOAPARP10MRGPRX4
SCHEMBL16808938 0.84 MAOB (0.61) MAOBMAOAIDO1MRGPRX4
SCHEMBL16795673 0.84 MAOB (0.69) MAOBMAOAIDO1AGXTPARP10
SCHEMBL2559064 0.83 ENPP2 (0.57) MAOBNR4A2MAOAPARP10MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515926-B1 FLUOROBENZAMIDES SUITABLE FOR THE TREATMENT OF ALZHEIMER'S DISEASE OR SENILE DEMENTIA HOFFMANN LA ROCHE (CH) 2009-04-08 EP disclosed
US-6951884-B2 Fluorobenzamides and uses thereof HOFFMANN-LA ROCHE INC. (US) 2005-10-04 US disclosed
EP-1515926-A2 FLUOROBENZAMIDES SUITABLE FOR THE TREATMENT OF ALZHEIMER'S DISEASE OR SENILE DEMENTIA F.HOFFMANN-LA ROCHE AG (CH) 2005-03-23 EP disclosed
US-20030236304-A1 Fluorobenzamides and uses thereof F. HOFFMANN-LA ROCHE AG (CH) 2003-12-25 US disclosed
WO-2003106380-A2 FLUOROBENZAMIDES F.HOFFMANN-LA ROCHE AG (CH) 2003-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030236304-A1 Fluorobenzamides and uses thereof MAOB, MAOA, BCHE MAOB 1/4885NR4A2 1698/4885MAOA 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.