SCHEMBL4427283

SCHEMBL4427283

COC(=O)c1ccc(C(c2cccc(F)c2)c2cccc(F)c2)[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
ALDH1A1 P00352 2/20 0.38
PARP1 P09874 1/20 0.38
ALOX5 P09917 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HSD17B2 P37059 2/20 0.37
HSD17B1 P14061 1/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4436626 0.84 CFTR (0.46) KDM4EGLAGAAALDH1A1MEN1
SCHEMBL4437347 0.84 GAA (0.51) KDM4EGLAGAAALDH1A1PARP1
SCHEMBL4439660 0.84 KDM4E (0.41) KDM4EGAAHDAC4HDAC7HDAC5
SCHEMBL4431487 0.84 KDM4E (0.54) KDM4EGLAGAAALDH1A1KMT2A
SCHEMBL4429591 0.79 GAA (0.51) KDM4EGLAGAAALDH1A1KMT2A
SCHEMBL4426018 0.77 KDM4E (0.49) KDM4EGLAGAAALDH1A1MEN1
SCHEMBL4438805 0.76 HSD17B2 (0.48) KDM4EGLAGAARAB9AHSD17B2
SCHEMBL4898553 0.75 KDM4E (0.60) KDM4EGLAGAAALDH1A1MAPT
SCHEMBL4428809 0.72 DAO (0.48) KDM4EGLAGAAALDH1A1MAPT
SCHEMBL4430946 0.71 HSD17B2 (0.46) KDM4EGAAALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed