SCHEMBL4436626

SCHEMBL4436626

COC(=O)c1ccc(C(c2cccc(C(F)(F)F)c2)c2cccc(C(F)(F)F)c2)[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.46
KDM4E B2RXH2 3/20 0.44
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
DAO P14920 1/20 0.44
GUSB P08236 1/20 0.43
KCNN4 O15554 1/20 0.40
CES2 O00748 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B2 P37059 3/20 0.39
MAPT P10636 2/20 0.39
LMNA P02545 3/20 0.39
RECQL P46063 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438805 0.85 HSD17B2 (0.48) CFTRKDM4EGLAGAAHSD17B2
SCHEMBL4427283 0.84 KDM4E (0.47) KDM4EGLAGAACES2HSD17B2
SCHEMBL4431487 0.81 KDM4E (0.54) CFTRKDM4EGLAGAANPSR1
SCHEMBL12427050 0.77 CFTR (0.52) CFTRKDM4EGLAGAAGUSB
SCHEMBL4429591 0.76 GAA (0.51) KDM4EGLAGAAHSD17B2MAPT
SCHEMBL4437347 0.76 GAA (0.51) KDM4EGLAGAAHSD17B2MAPT
SCHEMBL4898553 0.72 KDM4E (0.60) CFTRKDM4EGLAGAANPSR1
SCHEMBL4429494 0.70 KCNN4 (0.44) CFTRKDM4EKCNN4CES2NPSR1
SCHEMBL3056728 0.70 KDM4E (0.60) KDM4EGLAGAAHSD17B2
SCHEMBL6567957 0.69 CFTR (0.48) CFTRKDM4EGAAKCNN4CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed