SCHEMBL4437347

SCHEMBL4437347

COC(=O)c1ccc(C(c2ccc(F)cc2)c2ccc(F)cc2)[nH]c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.51
KDM4E B2RXH2 2/20 0.51
GLA P06280 1/20 0.51
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
RAB9A P51151 4/20 0.41
NPC1 O15118 3/20 0.41
CASP3 P42574 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4431487 0.86 KDM4E (0.54) GAAKDM4EGLASLC6A3RAB9A
SCHEMBL4438805 0.85 HSD17B2 (0.48) GAAKDM4EGLARAB9AHSD17B2
SCHEMBL4427283 0.84 KDM4E (0.47) GAAKDM4EGLARAB9ANPC1
SCHEMBL4429591 0.81 GAA (0.51) GAAKDM4EGLARAB9ACYP1A2
SCHEMBL4898553 0.79 KDM4E (0.60) GAAKDM4EGLASMN1; SMN2TSHR
SCHEMBL4426018 0.78 KDM4E (0.49) GAAKDM4EGLASLC6A4SLC6A3
SCHEMBL4436626 0.76 CFTR (0.46) GAAKDM4EGLASMN1; SMN2MEN1
SCHEMBL1547993 0.75 KDM4E (0.55) GAAKDM4EGLASLC6A4SLC6A3
SCHEMBL3913842 0.72 KDM4E (0.51) GAAKDM4EGLASLC6A4SLC6A3
SCHEMBL10464803 0.69 KDM4E (1.00) GAAKDM4EGLASMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed