Bicarbonate

Bicarbonate

SCHEMBL4428121

COc1cc(Cl)ccc1CC(=O)NC1CCC(C)CC1.O=C(O)O

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.66
MEN1 O00255 5/20 0.57
KMT2A Q03164 5/20 0.57
SIGMAR1 Q99720 3/20 0.49
LMNA P02545 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
TAS1R2 Q8TE23 1/20 0.46
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
LPAR1 Q92633 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL4424429 0.90 MEN1 (0.70) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4421056 0.89 MEN1 (0.56) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4421862 0.89 KMT2A (0.72) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4423971 0.89 KMT2A (0.72) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4434716 0.88 MEN1 (0.55) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4435083 0.88 MEN1 (0.55) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4435470 0.87 MEN1 (0.51) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4421083 0.87 MEN1 (0.54) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL4433274 0.86 MEN1 (0.56) GAAMEN1KMT2ASIGMAR1LMNA
Bicarbonate SCHEMBL7622161 0.85 SIGMAR1 (0.62) GAAMEN1KMT2ASIGMAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741700-B1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER CROPSCIENCE AG (DE) 2009-10-07 EP disclosed
EP-0741700-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AG (DE) 1996-11-13 EP disclosed
WO-1995020572-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1995-08-03 WO disclosed