SCHEMBL4428130

SCHEMBL4428130

O=C(O)c1ccc(C(c2ccccc2F)c2ccccc2F)[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
ALB P02768 1/20 0.37
NAPRT Q6XQN6 1/20 0.37
GAA P10253 3/20 0.36
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
NOTUM Q6P988 1/20 0.35
CNR2 P34972 1/20 0.35
KDM6B O15054 3/20 0.35
KDM4A O75164 3/20 0.35
KDM4D Q6B0I6 3/20 0.35
HIF1AN Q9NWT6 3/20 0.35
KDM5B Q9UGL1 3/20 0.35
KDM2A Q9Y2K7 3/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4426018 0.83 KDM4E (0.49) KDM4ECES2CES1GAAALDH1A1
SCHEMBL4431362 0.82 KDM4E (0.46) KDM4ENAPRTGAAALDH1A1KMT2A
SCHEMBL4427252 0.80 KDM4E (0.53) KDM4ENAPRTGAAALDH1A1KMT2A
SCHEMBL4439660 0.74 KDM4E (0.41) KDM4ECES2CES1NAPRTGAA
SCHEMBL3071414 0.74 KDM4E (0.49) KDM4ENAPRTGAAALDH1A1KMT2A
SCHEMBL5124119 0.71 KDM4E (0.49) KDM4ENAPRTGAAALDH1A1KDM6B
SCHEMBL4428254 0.70 HSD17B2 (0.49) KDM4ECES2CES1ALDH1A1KMT2A
SCHEMBL4429520 0.69 KDM4E (0.42) KDM4ENAPRTGAAALDH1A1LMNA
SCHEMBL4430946 0.69 HSD17B2 (0.46) KDM4EGAAALDH1A1KMT2ANOTUM
Phthalic Acid SCHEMBL3628215 0.65 CES2 (0.54) CES2CES1ALBGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed