SCHEMBL4429671

SCHEMBL4429671

CNCc1cn(S(=O)(=O)c2ccccc2CO)c(-c2cccnc2F)c1F

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
DHODH Q02127 2/20 0.33
ALOX5AP P20292 1/20 0.31
NAMPT P43490 2/20 0.31
CYP2C9 P11712 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
F10 P00742 1/20 0.31
FABP1 P07148 1/20 0.31
HTR6 P50406 2/20 0.30
CYP2D6 P10635 1/20 0.30
GRM4 Q14833 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1830844 0.88 DCTPP1 (0.33) NAMPTCYP2C9FABP1HTR6
SCHEMBL1580944 0.86 DCTPP1 (0.34) GRM4
SCHEMBL1580761 0.85 SLC40A1 (0.36) KDM4E
Hydrochloric Acid SCHEMBL2412383 0.85 DCTPP1 (0.33) GRM4
SCHEMBL1580308 0.85 HTR6 (0.41) NAMPTCYP2C9HTR6
Hydrochloric Acid SCHEMBL2415530 0.85 SLC40A1 (0.36) KDM4E
SCHEMBL1580925 0.84 L3MBTL1 (0.33) MAOAMAOBHTR6
SCHEMBL1580719 0.83 RXFP1 (0.31) HTR6
Fumaric Acid SCHEMBL1830756 0.83 DCTPP1 (0.33) DHODHNAMPTCYP2C9GRM4
Fumaric Acid SCHEMBL1830751 0.83 DCTPP1 (0.33) DHODHNAMPTCYP2C9GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed