SCHEMBL44301

SCHEMBL44301

COc1ccc(C(=O)NCc2cccc(-c3cn4ncccc4n3)c2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 9/20 0.66
GAA P10253 1/20 0.53
CHRM3 P20309 1/20 0.53
CYP3A4 P08684 2/20 0.53
ROCK2 O75116 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
PRKACA P17612 1/20 0.53
GSK3A P49840 1/20 0.53
GSK3B P49841 1/20 0.53
PRKX P51817 1/20 0.53
PRKCQ Q04759 1/20 0.53
ROCK1 Q13464 1/20 0.53
CLK4 Q9HAZ1 1/20 0.53
AURKA O14965 1/20 0.51
TP53 P04637 3/20 0.51
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13844942 0.87 WDR5 (0.52) WDR5CYP3A4ROCK2CYP2D6CYP2C9
SCHEMBL44512 0.87 WDR5 (0.52) WDR5GAACHRM3NPC1KDM4E
SCHEMBL44576 0.85 WDR5 (0.46) WDR5AURKAKDM4EALDH1A1
SCHEMBL44216 0.82 WDR5 (0.52) WDR5AURKANPC1RAB9AHPGD
SCHEMBL39537 0.82 WDR5 (0.46) WDR5KDM4EALDH1A1HPGDHSD17B10
SCHEMBL38703 0.82 WDR5 (0.44) WDR5ROCK2CYP2C9ROCK1AURKA
SCHEMBL19997605 0.79 WDR5 (1.00) WDR5
SCHEMBL44653 0.79 ALDH1A1 (0.54) WDR5GAACYP3A4KDM4EALDH1A1
SCHEMBL12951391 0.78 WDR5 (0.41) WDR5GAACYP3A4ROCK2CYP2D6
SCHEMBL13844884 0.78 WDR5 (0.41) WDR5GAACYP3A4ROCK2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed