SCHEMBL4430613

SCHEMBL4430613

CCCCC(C(=O)N[C@@H](CC(=O)O)c1ccc(C)cc1)n1cc(C)cc(Cc2ccc3ccccc3c2)c1=O

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSA P10619 3/20 0.40
KEAP1 Q14145 2/20 0.38
NFE2L2 Q16236 2/20 0.38
CASP1 P29466 11/20 0.38
BDKRB2 P30411 1/20 0.38
FPR1 P21462 2/20 0.35
CYP26A1 O43174 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4426794 0.97 CASP1 (0.39) CTSACASP1BDKRB2FPR1
SCHEMBL8506622 0.93 CTSA (0.40) CTSAKEAP1NFE2L2FPR1CYP26A1
SCHEMBL4435400 0.93 CTSA (0.40) CTSAKEAP1NFE2L2FPR1CYP26A1
SCHEMBL4435399 0.93 CTSA (0.40) CTSAKEAP1NFE2L2FPR1CYP26A1
SCHEMBL4431712 0.90 CTSA (0.41) CTSAKEAP1NFE2L2FPR1CYP26A1
SCHEMBL4436967 0.90 CTSA (0.41) CTSAKEAP1NFE2L2FPR1CYP26A1
SCHEMBL4431319 0.90 KEAP1 (0.43) KEAP1NFE2L2CASP1FPR1
SCHEMBL4436767 0.89 CASP1 (0.39) CASP1FPR1
SCHEMBL4425710 0.89 ALDH1A1 (0.37) CTSAKEAP1NFE2L2FPR1
SCHEMBL4426449 0.89 CYP26A1 (0.39) CTSAKEAP1NFE2L2FPR1CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1213288-B1 Propanoic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2009-01-14 EP disclosed
EP-1213288-A1 Propanoic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-06-12 EP disclosed