SCHEMBL4436967

SCHEMBL4436967

CCCCC(C(=O)N[C@@H](CC(=O)O)c1ccc(-c2ccc(C)cc2)cc1)n1cc(C)cc(Cc2ccccc2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSA P10619 8/20 0.41
CYP26A1 O43174 1/20 0.36
KEAP1 Q14145 2/20 0.35
NFE2L2 Q16236 2/20 0.35
UTS2R Q9UKP6 3/20 0.35
FPR1 P21462 2/20 0.34
MMP2 P08253 2/20 0.34
MMP1 P03956 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4431712 1.00 CTSA (0.41) CTSACYP26A1KEAP1NFE2L2UTS2R
SCHEMBL4435258 0.97 CTSA (0.41) CTSAFPR1MMP2MMP1
SCHEMBL4435400 0.97 CTSA (0.40) CTSACYP26A1KEAP1NFE2L2UTS2R
SCHEMBL4435399 0.97 CTSA (0.40) CTSACYP26A1KEAP1NFE2L2UTS2R
SCHEMBL8506622 0.97 CTSA (0.40) CTSACYP26A1KEAP1NFE2L2UTS2R
SCHEMBL4427187 0.94 MMP2 (0.38) CTSAFPR1MMP2MMP1
SCHEMBL7429087 0.94 MMP2 (0.38) CTSAFPR1MMP2MMP1
SCHEMBL4426400 0.93 CYP26A1 (0.38) CTSACYP26A1FPR1MMP2MMP1
SCHEMBL4435266 0.93 FPR1 (0.40) CTSACYP26A1FPR1
SCHEMBL4425710 0.92 ALDH1A1 (0.37) CTSAKEAP1NFE2L2FPR1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1213288-B1 Propanoic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2009-01-14 EP disclosed
EP-1213288-A1 Propanoic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-06-12 EP disclosed