SCHEMBL4430631

SCHEMBL4430631

O=C(O)c1c(C(c2cccc(C(F)(F)F)c2)c2cccc(C(F)(F)F)c2)cc[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 2/20 0.42
CES2 O00748 2/20 0.42
DAO P14920 1/20 0.41
PNMT P11086 1/20 0.39
ALKBH5 Q6P6C2 1/20 0.38
SRD5A2 P31213 1/20 0.38
MAOB P27338 1/20 0.38
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
HSD11B1 P28845 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KMO O15229 1/20 0.36
PARP1 P09874 1/20 0.36
EPHX1 P07099 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6821850 0.72 DAO (0.48) ACP3DAOMEN1KMT2A
SCHEMBL4086256 0.72 PNMT (0.58) ACP3CES2DAOPNMTIDO1
SCHEMBL13357679 0.71 IDO1 (0.59) ACP3CES2PNMTIDO1TDO2
SCHEMBL18952889 0.67 CES2 (0.57) ACP3CES2PNMTSRD5A2IDO1
SCHEMBL4437624 0.66 DAO (0.47) ACP3CES2DAOPNMTSRD5A2
SCHEMBL5159944 0.66 CES2 (0.69) ACP3CES2PNMTSRD5A2IDO1
SCHEMBL6674012 0.66 CES2 (0.69) ACP3CES2PNMTSRD5A2IDO1
SCHEMBL7436009 0.66 CES2 (0.55) ACP3CES2PNMTSRD5A2IDO1
SCHEMBL5159938 0.66 CES2 (0.69) ACP3CES2PNMTSRD5A2IDO1
SCHEMBL15019153 0.66 CES2 (0.55) ACP3CES2PNMTSRD5A2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed