SCHEMBL4430755

SCHEMBL4430755

C=CN1CCN(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.53
CA2 P00918 2/20 0.51
CA9 Q16790 2/20 0.51
CA12 O43570 1/20 0.51
DHFR P00374 1/20 0.46
ME2 P23368 1/20 0.43
ME1 P48163 1/20 0.43
ME3 Q16798 1/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
PHGDH O43175 1/20 0.43
MLYCD O95822 1/20 0.43
CACNA1G O43497 1/20 0.42
DRD4 P21917 1/20 0.42
GRM2 Q14416 1/20 0.42
NOTUM Q6P988 1/20 0.42
MAOB P27338 1/20 0.42
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28650484 0.84 CA12 (0.65) AKR1C3CA2CA9CA12DHFR
SCHEMBL13632333 0.82 AKR1C3 (0.56) AKR1C3CA2CA9CA12DHFR
SCHEMBL4432185 0.79 LMNA (0.57) AKR1C3CA2CA9CA12CA1
SCHEMBL4434038 0.78 KCNA5 (0.47)
SCHEMBL28818468 0.78 AKR1C3 (0.52) AKR1C3CA2CA9CA12DHFR
SCHEMBL21583753 0.77 CA12 (0.66) AKR1C3CA2CA9CA12ME2
SCHEMBL13285321 0.77 CA12 (0.56) AKR1C3CA2CA9CA12DHFR
SCHEMBL28842325 0.77 CA12 (0.56) AKR1C3CA2CA9CA12DHFR
SCHEMBL2750409 0.77 MAPT (0.50) AKR1C3PHGDHDRD4HTR1ADRD2
SCHEMBL21180901 0.76 CYP3A4 (0.52) AKR1C3CA2CA9CA12DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090156612-A1 Substituted imidazole compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156612-A1 Substituted imidazole compound and use thereof REN, ACE, AGT AKR1C3 156/4885CA2 218/4885CA9 209/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.