SCHEMBL21180901

SCHEMBL21180901

C=CC1CCN(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.52
NOTUM Q6P988 1/20 0.50
HRH4 Q9H3N8 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
CA12 O43570 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
AKR1C3 P42330 1/20 0.43
DEGS1 O15121 1/20 0.42
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
DHFR P00374 1/20 0.40
MAOB P27338 3/20 0.40
GPR119 Q8TDV5 1/20 0.40
ME2 P23368 1/20 0.39
ME1 P48163 1/20 0.39
ME3 Q16798 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12419722 0.83 NOTUM (0.54) CYP3A4NOTUMHRH4HRH3CA12
SCHEMBL2093736 0.81 NOTUM (0.54) CYP3A4NOTUMHRH4HRH3CA12
SCHEMBL28650484 0.78 CA12 (0.65) CYP3A4NOTUMHRH4HRH3CA12
SCHEMBL21180882 0.77 ADRB1 (0.48) AKR1C3GPR119
SCHEMBL1704614 0.77 NOTUM (0.54) CYP3A4NOTUMHRH4HRH3CA12
SCHEMBL2056103 0.77 NOTUM (0.54) CYP3A4NOTUMHRH4HRH3CA12
SCHEMBL61425 0.77 NOTUM (0.58) CYP3A4NOTUMHRH4HRH3CA12
SCHEMBL26143961 0.77 MBTD1 (0.52) CYP3A4NOTUM
Hydrochloric Acid SCHEMBL5220023 0.76 NOTUM (0.53) CYP3A4NOTUMHRH4HRH3CA12
SCHEMBL4430755 0.76 AKR1C3 (0.53) CYP3A4NOTUMCA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3221304-B1 NOVEL CARBOXYLIC ACID COMPOUNDS USEFUL FOR INHIBITING MICROSOMAL PROSTAGLANDIN E2 SYNTHASE-1 LILLY CO ELI (US) 2019-07-24 EP disclosed