SCHEMBL4432302

SCHEMBL4432302

COC(=O)C1CCc2ccccc2C1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 4/20 0.53
MTNR1B P49286 4/20 0.53
FAAH O00519 7/20 0.51
GHSR Q92847 1/20 0.50
P2RX7 Q99572 1/20 0.47
KMT2A Q03164 1/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
HSD11B1 P28845 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29882799 1.00 MTNR1A (0.53) MTNR1AMTNR1BFAAHGHSRP2RX7
SCHEMBL29519648 0.87 KMT2A (0.54) MTNR1AMTNR1BFAAHKMT2AHSD11B1
SCHEMBL857083 0.87 KMT2A (0.54) MTNR1AMTNR1BFAAHKMT2AHSD11B1
SCHEMBL31330957 0.83 FAAH (0.49) MTNR1AMTNR1BFAAHGHSRP2RX7
SCHEMBL12473133 0.82 FAAH (0.63) FAAH
SCHEMBL10260957 0.82 FAAH (0.57) FAAH
SCHEMBL30437453 0.82 KDM4E (0.50) MTNR1AMTNR1BFAAHGHSRKMT2A
SCHEMBL3630406 0.82 KDM4E (0.50) MTNR1AMTNR1BFAAHGHSRKMT2A
SCHEMBL6819517 0.82 MTNR1A (0.64) MTNR1AMTNR1B
SCHEMBL8074265 0.82 MTNR1A (0.64) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1069309-C N-(3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphtalene-2-carboxamide derivative, preparation and application of same SANNOFFE SYNTHELABO (FR) 2001-08-08 CN claimed
CN-1109870-A N-(3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphtalene-2-carboxamide derivative, preparation and application of same SYNTHELABO (FR) 1995-10-11 CN claimed
CN-115197036-B Method for performing anti-mahalanobis hydrogen carboxylation reaction on photocatalytic olefin compound and carbon dioxide 中国科学院理化技术研究所 2024-01-23 CN disclosed
CN-115197036-A Method for carrying out anti-Ma hydrocarboxylation reaction on olefin compound and carbon dioxide by photocatalysis 中国科学院理化技术研究所 2022-10-18 CN disclosed
CN-106687446-B 5-amino-4-carbamoyl-pyrazole compounds as selective and irreversible kinase inhibitors of T790M/WT-EGFR and uses thereof 百济神州(北京)生物科技有限公司 2020-04-28 CN disclosed
CN-104583177-B Aryl alkyl amines as calcium-sensing receptor regulator 卢平亚特兰蒂斯控股有限公司 2016-09-07 CN disclosed
WO-2016008411-A1 5-AMINO-4-CARBAMOYL-PYRAZOLE COMPOUNDS AS SELECTIVE AND IRREVERSIBLE T790M OVER WT-EGFR KINASE INHIBITORS AND USE THEREOF BEIGENE, LTD. (KY) 2016-01-21 WO disclosed
US-9163001-B2 Substituted chroman compounds as calcium sensing receptor modulators LUPIN LIMITED (IN) 2015-10-20 US disclosed
US-9163001-B2 Substituted chroman compounds as calcium sensing receptor modulators LUPIN LIMITED (IN) 2015-10-20 US disclosed
CN-104583177-A Arylalkylamine compounds as calcium sensing receptor modulators LUPIN LTD 2015-04-29 CN disclosed
US-20150038546-A1 SUBSTITUTED CHROMAN COMPOUNDS AS CALCIUM SENSING RECEPTOR MODULATORS LUPIN LIMITED (IN) 2015-02-05 US disclosed
EP-0516980-B1 Novel 2-mercaptomethylene-tetrahydronaphthalene and indane-2-carboxamide derivatives as enkephalinase inhibitors MERRELL PHARMA INC (US) 1996-04-17 EP disclosed
CN-1109870-A N-(3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphtalene-2-carboxamide derivative, preparation and application of same SYNTHELABO (FR) 1995-10-11 CN disclosed
US-5252601-A 2-mercaptomethylene-tetrahydronaphthalene and indane-2-carboxamide derivatives as enkephalinase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed
EP-0310745-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ORION-YHTYMÄ OY (FI) 1993-01-27 EP disclosed
EP-0516980-A1 Novel 2-mercaptomethylene-tetrahydronaphthalene and indane-2-carboxamide derivatives as enkephalinase inhibitors MERRELL PHARMACEUTICALS INC. (US) 1992-12-09 EP disclosed
EP-0183492-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Farmos-Yhtyma Oy (FI) 1989-11-15 EP disclosed
EP-0310745-A2 Substituted imidazole derivatives and their preparation and use ORION-YHTYMÄ OY (FI) 1989-04-12 EP disclosed
US-4689339-A 4-dihydroinden-2-yl-, 4-tetrahydronaphth-2-yl-, and 4-dihydrobenzofuran-2-ylimidazoles, useful to block α2 -adrenergic receptors FARMOS YHTYMA OY (FI) 1987-08-25 US disclosed
EP-0183492-A1 Substituted imidazole derivatives and their preparation and use Farmos-Yhtyma Oy (FI) 1986-06-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150038546-A1 SUBSTITUTED CHROMAN COMPOUNDS AS CALCIUM SENSING RECEPTOR MODULATORS CASR, RYR2, CALCR MTNR1A 135/4885MTNR1B 340/4885FAAH 3844/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.