SCHEMBL857083

SCHEMBL857083

COC(=O)C1Cc2ccccc2C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
BUB1 O43683 1/20 0.46
ALDH1A1 P00352 2/20 0.45
FAAH O00519 1/20 0.45
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
BRD4 O60885 1/20 0.43
MEN1 O00255 1/20 0.43
HSD11B1 P28845 1/20 0.42
TSHR P16473 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NPY5R Q15761 1/20 0.42
POLB P06746 1/20 0.42
GRM7 Q14831 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29519648 1.00 KMT2A (0.54) KMT2ABUB1ALDH1A1FAAHMTNR1A
SCHEMBL29882799 0.87 MTNR1A (0.53) KMT2AALDH1A1FAAHMTNR1AMTNR1B
SCHEMBL4432302 0.87 MTNR1A (0.53) KMT2AALDH1A1FAAHMTNR1AMTNR1B
SCHEMBL15519819 0.84 KMT2A (0.56) KMT2ABUB1ALDH1A1BRD4TSHR
SCHEMBL8911487 0.84 KMT2A (0.56) KMT2ABUB1ALDH1A1BRD4TSHR
SCHEMBL17540272 0.83 KMT2A (0.44) KMT2ABUB1ALDH1A1HSD11B1TSHR
SCHEMBL12472574 0.82 FAAH (0.55) KMT2AFAAHNPY5R
SCHEMBL1339793 0.81 KMT2A (0.46) KMT2AMTNR1AMTNR1BMEN1SMN1; SMN2
SCHEMBL31278113 0.81 KMT2A (0.46) KMT2ABUB1ALDH1A1MTNR1AMTNR1B
SCHEMBL9979464 0.81 CA1 (0.46) KMT2AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 160 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002002119-A1 FATTY ACID SYNTHASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-01-10 WO claimed
US-12559455-B2 Compound as a UBR box domain ligand AUTOTAC INC. (KR) 2026-02-24 US disclosed
US-20250326764-A1 INHIBITORS OF THE MENIN-MLL INTERACTION VITAE PHARMACEUTICALS LLC (US) 2025-10-23 US disclosed
US-12312359-B2 Inhibitors of the menin-MLL interaction VITAE PHARMACEUTICALS, LLC (US) 2025-05-27 US disclosed
US-12286411-B2 Indane derivatives for use in the treatment of bacterial infection ANTABIO SAS (FR) 2025-04-29 US disclosed
US-12247013-B2 Indane derivatives for use in the treatment of bacterial infection ANTABIO SAS (FR) 2025-03-11 US disclosed
WO-2024163752-A1 HETEROCYCLIC COMPOUNDS AS PI3Kα INHIBITORS SYNNOVATION THERAPEUTICS, INC. (US) 2024-08-08 WO disclosed
EP-4408416-A1 ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE Petra Pharma Corporation (US) 2024-08-07 EP disclosed
US-12030862-B2 Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of disease PETRA PHARMA CORPORATION (US) 2024-07-09 US disclosed
US-12030862-B2 Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of disease PETRA PHARMA CORPORATION (US) 2024-07-09 US disclosed
US-4689339-A 4-dihydroinden-2-yl-, 4-tetrahydronaphth-2-yl-, and 4-dihydrobenzofuran-2-ylimidazoles, useful to block α2 -adrenergic receptors FARMOS YHTYMA OY (FI) 1987-08-25 US disclosed
EP-0183492-A1 Substituted imidazole derivatives and their preparation and use Farmos-Yhtyma Oy (FI) 1986-06-04 EP disclosed
EP-0056271-B1 CARBOXYLIC ACID ESTERS AND INSECTICIDAL AND/OR ACARICIDAL COMPOSITIONS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1986-05-07 EP disclosed
US-4559356-A ANTIDE PRESSANTS; HYPERTENSIVE AGENTS SYNTHELABO (FR) 1985-12-17 US disclosed
US-4480118-A Carboxylic acid ester and an insecticidal and/or acaricidal composition containing the same SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1984-10-30 US disclosed
EP-0056271-A2 Carboxylic acid esters and insecticidal and/or acaricidal compositions SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1982-07-21 EP disclosed
US-4269848-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETICS LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1981-05-26 US disclosed
US-4224341-A ANTIINFLAMMATORY AGENTS, ANALGESICS AND ANTIPYRETICS LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1980-09-23 US disclosed
US-4166131-A ANTIINFLAMMATORY AGENTS, ANTIPYRETICS, ANTIARTHRITIC AGENT HEXACHIMIE SOCIETE ANONYME (FR) 1979-08-28 US disclosed
US-4152527-A 15-Substituted-ω-pentanorprostaglandins PFIZER INC. (US) 1979-05-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12286411-B2 Indane derivatives for use in the treatment of bacterial infection ELANE, ARG1, INSRR KMT2A 3671/4885BUB1 908/4885ALDH1A1 1376/4885
US-12312359-B2 Inhibitors of the menin-MLL interaction MLLT1, MEN1, MLLT3 KMT2A 12/4885BUB1 661/4885ALDH1A1 4369/4885
US-12030862-B2 Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of disease PIK3CA, PIK3R4, PIK3R5 KMT2A 4426/4885BUB1 1179/4885ALDH1A1 3412/4885
US-12559455-B2 Compound as a UBR box domain ligand UBR4, UBTF, UBQLN1 KMT2A 574/4885BUB1 2220/4885ALDH1A1 1486/4885
US-12247013-B2 Indane derivatives for use in the treatment of bacterial infection ELANE, ARG1, INSRR KMT2A 3671/4885BUB1 908/4885ALDH1A1 1376/4885
US-20250326764-A1 INHIBITORS OF THE MENIN-MLL INTERACTION MLLT1, MEN1, MLLT3 KMT2A 12/4885BUB1 661/4885ALDH1A1 4369/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.