SCHEMBL4432793

SCHEMBL4432793

COCC1c2sc(OC(=O)OC)cc2CCN1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN2 Q9H2S1 4/20 0.34
KCNN3 Q9UGI6 4/20 0.34
KCNN1 Q92952 2/20 0.34
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GRIN2D O15399 8/20 0.32
GRIN3B O60391 8/20 0.32
GRIN1 Q05586 8/20 0.32
GRIN2A Q12879 8/20 0.32
GRIN2B Q13224 8/20 0.32
GRIN2C Q14957 8/20 0.32
GRIN3A Q8TCU5 8/20 0.32
OPRM1 P35372 3/20 0.32
OPRK1 P41145 3/20 0.32
KCNH2 Q12809 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
OPRL1 P41146 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13372740 0.89 KCNN2 (0.34) KCNN2KCNN3KCNN1GRIN2DGRIN3B
SCHEMBL13372899 0.83 MAOA (0.39) HTTSMN1; SMN2ALDH1A1POLB
SCHEMBL3307517 0.81 KDM4E (0.40) KCNN2KCNN3KCNN1HTTSMN1; SMN2
SCHEMBL3303694 0.79 KDM4E (0.36) KCNN2KCNN3KCNN1KDM4EALDH1A1
SCHEMBL4440893 0.77 CYP3A4 (0.31) SMN1; SMN2
SCHEMBL3305816 0.76 KCNN2 (0.39) KCNN2KCNN3KCNN1OPRK1KDM4E
SCHEMBL4582601 0.71 ALDH1A1 (0.38) OPRM1KDM4EALDH1A1POLB
SCHEMBL4431441 0.69 WDR91 (0.41) KDM4EALDH1A1
SCHEMBL4428221 0.69 MAOA (0.40) SMN1; SMN2ALDH1A1
SCHEMBL3311778 0.67 KCNN2 (0.38) KCNN2KCNN3KCNN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132193-B1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INT (DE) 2012-10-24 EP disclosed
EP-2132193-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS Boehringer Ingelheim International GmbH (DE) 2009-12-16 EP disclosed
WO-2008116881-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-02 WO disclosed