SCHEMBL4432979

SCHEMBL4432979

COc1ccc(C(C(C)=O)c2cccc(C(F)(F)F)c2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.51
AKR1C2 P52895 3/20 0.51
CMA1 P23946 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.46
LMNA P02545 3/20 0.46
NQO2 P16083 1/20 0.46
KDM4E B2RXH2 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
POLB P06746 1/20 0.44
CES2 O00748 1/20 0.44
MAPT P10636 1/20 0.43
HTT P42858 2/20 0.43
SOS1 Q07889 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KRAS P01116 1/20 0.42
SCD O00767 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4434628 0.88 AKR1C3 (0.51) AKR1C3AKR1C2MAPT
SCHEMBL4438527 0.83 CES2 (0.50) AKR1C3AKR1C2SMN1; SMN2POLBCES2
SCHEMBL11103452 0.82 ACP3 (0.55) SMN1; SMN2POLBCES2MAPTHTT
SCHEMBL16973606 0.82 TDP1 (0.51) SMN1; SMN2LMNATDP1POLBMAPT
SCHEMBL8295353 0.81 NR1H4 (0.45) SMN1; SMN2LMNAKDM4ETDP1NPSR1
SCHEMBL4432351 0.80 AKR1C3 (0.49) AKR1C3AKR1C2SMN1; SMN2MAPTNPSR1
SCHEMBL4436028 0.80 AKR1C3 (0.49) AKR1C3AKR1C2NPSR1
SCHEMBL4430282 0.77 PDE10A (0.46) AKR1C3AKR1C2LMNANPSR1
SCHEMBL4430480 0.76 AKR1C3 (0.48) AKR1C3AKR1C2LMNAKDM4EMAPT
SCHEMBL4432347 0.76 ALDH1A1 (0.50) LMNAKDM4EPOLBMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed