SCHEMBL4433860

SCHEMBL4433860

O=C(O)Oc1ccc2ccc3[nH]ncc3cc1-2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.49
CLK1 P49759 2/20 0.49
CLK2 P49760 2/20 0.49
CDK5 Q00535 2/20 0.49
DYRK1A Q13627 2/20 0.49
CLK4 Q9HAZ1 2/20 0.49
DYRK1B Q9Y463 2/20 0.49
DYRK3 O43781 1/20 0.49
CLK3 P49761 1/20 0.49
CDK5R1 Q15078 1/20 0.49
DYRK2 Q92630 1/20 0.49
TRPA1 O75762 6/20 0.44
ROCK2 O75116 4/20 0.44
ROCK1 Q13464 3/20 0.44
TLR8 Q9NR97 1/20 0.44
CTNNB1 P35222 1/20 0.44
WNT3A P56704 1/20 0.44
JAK2 O60674 3/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6574033 0.77 RAB9A (0.49) GSK3BCLK1CLK2CDK5DYRK1A
SCHEMBL31253099 0.70 GSK3B (0.68) GSK3BCLK1CLK2CDK5DYRK1A
SCHEMBL23063810 0.70 GSK3B (0.68) GSK3BCLK1CLK2CDK5DYRK1A
SCHEMBL2192642 0.69 TRPA1 (0.40) TRPA1ROCK1CTNNB1WNT3ANPC1
SCHEMBL261380 0.68 CTNNB1 (0.65) GSK3BCLK1CLK2CDK5DYRK1A
SCHEMBL30270547 0.68 CTNNB1 (0.65) GSK3BCLK1CLK2CDK5DYRK1A
SCHEMBL17697651 0.68 SLC6A9 (0.51) NPC1RAB9A
SCHEMBL4039954 0.68 FGFR1 (0.47) CLK2DYRK1ACLK4NPC1RAB9A
Hydrochloric Acid SCHEMBL1665151 0.67 CTNNB1 (0.63) GSK3BCLK1CLK2CDK5DYRK1A
SCHEMBL27556162 0.67 PTGDR2 (0.54) MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2094711-A1 STRUCTURAL MIMETICS OF PROLINE-RICH PEPTIDES AND THE PHARMACEUTICAL USE THEREOF Forschungsverbund Berlin e.V. (DE) 2009-09-02 EP disclosed
WO-2008040332-A1 STRUCTURAL MIMETICS OF PROLINE-RICH PEPTIDES AND THE PHARMACEUTICAL USE THEREOF FORSCHUNGSVERBUND BERLIN E.V. (DE) 2008-04-10 WO disclosed