SCHEMBL4434660

SCHEMBL4434660

Cc1cc([C@H](CCN[C@@H](C(N)=O)c2ccccc2)c2ccc(C(F)(F)F)cc2)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 4/20 0.43
EPHX2 P34913 4/20 0.43
TACR1 P25103 1/20 0.41
TACR3 P29371 1/20 0.41
CCR2 P41597 3/20 0.41
ALDH1A1 P00352 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
CNR2 P34972 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HAT1 O14929 2/20 0.39
EP300 Q09472 2/20 0.39
CNR1 P21554 2/20 0.39
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 3/20 0.38
NPC1 O15118 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 2/20 0.38
MTOR P42345 2/20 0.38
RAB9A P51151 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4427996 1.00 ALOX5 (0.43) ALOX5EPHX2TACR1TACR3CCR2
SCHEMBL4432435 0.89 CNR1 (0.49) ALDH1A1CNR2CNR1SLC6A2SLC6A4
SCHEMBL4441795 0.88 KDM4E (0.46) ALOX5EPHX2TACR1TACR3CCR2
SCHEMBL4430647 0.88 KDM4E (0.46) ALOX5EPHX2TACR1TACR3CCR2
SCHEMBL4432382 0.86 ALOX5 (0.39) ALOX5EPHX2TACR1TACR3CCR2
SCHEMBL4431479 0.86 ALOX5 (0.39) ALOX5EPHX2TACR1TACR3CCR2
SCHEMBL4434471 0.85 CNR1 (0.43) ALDH1A1CNR2CNR1SLC6A3CYP2C19
SCHEMBL4430509 0.85 P2RX7 (0.44) EPHX2EP300LMNA
SCHEMBL4432823 0.85 P2RX7 (0.44) EPHX2EP300LMNA
SCHEMBL4429659 0.85 P2RX7 (0.44) EPHX2EP300LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed