SCHEMBL4436057

SCHEMBL4436057

CC(=O)C(c1ccc(C(F)(F)F)cc1)c1ccc2nc(C)sc2c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.48
LDHA P00338 1/20 0.46
PPARA Q07869 1/20 0.43
ALDH1A1 P00352 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
HTT P42858 2/20 0.42
CSNK1D P48730 1/20 0.41
MAPT P10636 3/20 0.41
EPHX2 P34913 1/20 0.41
SCN4A P35499 1/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 3/20 0.40
CYP2D6 P10635 1/20 0.39
MEN1 O00255 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
ACP1 P24666 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4432461 0.77 AHR (0.39) DYRK1AALDH1A1NPC1MAPTKMT2A
SCHEMBL11956363 0.77 EPHX2 (0.65) DYRK1ALDHAPPARAALDH1A1TDP1
SCHEMBL4431654 0.76 ALDH1A1 (0.48) DYRK1AALDH1A1SMN1; SMN2MAPT
SCHEMBL4432335 0.74 CES2 (0.41) PPARAMAPTTP53
SCHEMBL23932781 0.74 LDHA (0.52) LDHAALDH1A1TDP1NPC1RAB9A
SCHEMBL4432365 0.72 AKR1C3 (0.43) PPARAALDH1A1
SCHEMBL12109822 0.72 MAPT (0.38) DYRK1AALDH1A1TDP1NPC1RAB9A
SCHEMBL4431561 0.72 AKR1C3 (0.48) ALDH1A1
SCHEMBL4438527 0.72 CES2 (0.50) ALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL4435426 0.71 CNR1 (0.40) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed