SCHEMBL4432461

SCHEMBL4432461

CC(=O)C(c1ccc(C(F)(F)F)cc1)c1sc(C)nc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
POLB P06746 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
FFAR1 O14842 1/20 0.37
CDK2 P24941 1/20 0.37
PDE2A O00408 4/20 0.37
HSD11B1 P28845 1/20 0.36
NTRK1 P04629 1/20 0.35
DYRK1A Q13627 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CRHBP P24387 1/20 0.35
KMT2A Q03164 1/20 0.35
CRHR2 Q13324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4436057 0.77 DYRK1A (0.48) NPC1ALDH1A1DYRK1AMAPTMEN1
SCHEMBL2304585 0.71 ACP3 (0.56) NPC1ALDH1A1CES2CES1HSD11B1
SCHEMBL4435804 0.71 HSD11B1 (0.45) CES2CES1PDE2AHSD11B1
SCHEMBL4435069 0.70 CES2 (0.41) NPC1ALDH1A1CES2CES1FFAR1
SCHEMBL4432335 0.70 CES2 (0.41) CES2CES1PDE2AMAPT
SCHEMBL4436009 0.69 MEN1 (0.43) ALDH1A1CES2CES1PDE2AHSD11B1
SCHEMBL4433211 0.69 LMNA (0.41) NPC1ALDH1A1CES2CES1PDE2A
SCHEMBL4434570 0.69 FFAR1 (0.44) NPC1ALDH1A1CES2CES1FFAR1
SCHEMBL4432365 0.68 AKR1C3 (0.43) ALDH1A1CES2CES1PDE2A
SCHEMBL4431036 0.68 KCNQ3 (0.51) ALDH1A1CES2CES1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed