SCHEMBL4437241

SCHEMBL4437241

O=CC(O)C1(c2cccs2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.45
SLC6A4 P31645 1/20 0.43
OPRM1 P35372 2/20 0.37
OPRL1 P41146 2/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
SLC6A2 P23975 1/20 0.37
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
PRCP P42785 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14857042 0.66 SLC6A2 (0.47) SLC6A3SLC6A4OPRM1OPRL1OPRD1
SCHEMBL1308581 0.65
SCHEMBL4446504 0.64 MAOA (0.39) SLC6A3SLC6A4OPRM1OPRL1OPRD1
SCHEMBL14856965 0.64 SLC6A2 (0.50) SLC6A3SLC6A4OPRM1OPRL1SLC6A2
SCHEMBL4438204 0.64 CYP2A6 (0.34) SLC6A3OPRM1OPRL1OPRD1OPRK1
SCHEMBL2795442 0.63 ALDH1A1 (0.51) OPRM1OPRL1KMT2AMEN1ALDH1A1
SCHEMBL5263610 0.62 ALDH1A1 (0.47) KMT2AALDH1A1LMNATP53HTT
SCHEMBL3521022 0.62 SLC6A3 (1.00) SLC6A3SLC6A4SLC6A2KMT2AMEN1
SCHEMBL1309560 0.62 OPRM1 (0.54) SLC6A3SLC6A4OPRM1OPRL1OPRD1
SCHEMBL1310931 0.62 OPRM1 (0.54) SLC6A3SLC6A4OPRM1OPRL1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134692-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION Wyeth a Corporation of the State of Delaware (US) 2009-12-23 EP disclosed
WO-2008121817-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION WYETH (US) 2008-10-09 WO disclosed