SCHEMBL4437705

SCHEMBL4437705

CCOC(=O)C1CCC(c2cc(F)c(F)c(F)c2)N1C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.39
ALDH1A1 P00352 4/20 0.37
TYMS P04818 1/20 0.37
TSHR P16473 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GPR119 Q8TDV5 4/20 0.35
TDP1 Q9NUW8 1/20 0.34
RIPK1 Q13546 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
PDE5A O76074 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2351664 1.00 DPP4 (0.39) DPP4ALDH1A1TYMSTSHRKDM4E
SCHEMBL2346142 0.90 ALDH1A1 (0.43) DPP4ALDH1A1TYMSTSHRKDM4E
SCHEMBL2587508 0.90 FFAR2 (0.38) DPP4ALDH1A1TYMSTSHRKDM4E
SCHEMBL3589461 0.85 TYMS (0.41) ALDH1A1TYMSGPR119TDP1MEN1
SCHEMBL2351853 0.85 TYMS (0.41) ALDH1A1TYMSGPR119TDP1MEN1
SCHEMBL4441921 0.85 TYMS (0.41) ALDH1A1TYMSGPR119TDP1MEN1
SCHEMBL20835401 0.85 TYMS (0.35) DPP4ALDH1A1TYMSTSHRKDM4E
SCHEMBL2587662 0.84 DPP4 (0.41) DPP4ALDH1A1TYMSTSHRKDM4E
SCHEMBL20835437 0.84 L3MBTL1 (0.41) DPP4ALDH1A1TYMSTSHRKDM4E
SCHEMBL2584143 0.84 RIPK1 (0.46) ALDH1A1TYMSGPR119TDP1RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125829-A2 BICYCLIC OXOMORPHOLINE DERIVATIVE Eisai R&D Management Co., Ltd. (JP) 2009-12-02 EP disclosed
WO-2008108378-A2 BICYCLIC OXOMORPHOLINE DERIVATIVE EISAI R & D MANAGEMENT CO., LTD. (JP) 2008-09-12 WO disclosed