SCHEMBL4437800

SCHEMBL4437800

O=C(O)CCc1c(C(=O)c2ccc(Cl)cc2)oc2cc(O)ccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 2/20 0.52
HPGD P15428 2/20 0.52
GLA P06280 1/20 0.52
GAA P10253 1/20 0.52
TSHR P16473 1/20 0.52
CASP1 P29466 1/20 0.52
CASP7 P55210 1/20 0.52
HSD17B10 Q99714 1/20 0.52
NPSR1 Q6W5P4 3/20 0.47
MAPT P10636 3/20 0.47
HTT P42858 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
ALOX12 P18054 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ESR1 P03372 2/20 0.47
ESR2 Q92731 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
LMNA P02545 2/20 0.45
NPC1 O15118 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12013388 0.89 HTT (0.47) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL8543822 0.88 CASP1 (0.52) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL8544863 0.88 KDM4E (0.58) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL8550054 0.87 SLC22A12 (0.44) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL8308344 0.87 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL679245 0.86 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL8837860 0.86 KDM4E (0.52) ALDH1A1KDM4EHPGDGLAGAA
SCHEMBL8551230 0.84 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDNPSR1MAPT
SCHEMBL5964314 0.83 HTT (0.46) ALDH1A1KDM4EHPGDNPSR1MAPT
SCHEMBL8307013 0.82 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2068872-A1 COMBINATIONS CONTAINING A 4-ACYLAMINOPYRIDINE DERIVATIVE Braincells, Inc. (US) 2009-06-17 EP disclosed
WO-2008030651-A1 COMBINATIONS CONTAINING A 4-ACYLAMINOPYRIDINE DERIVATIVE BRAINCELLS, INC. (US) 2008-03-13 WO disclosed