SCHEMBL8308344

SCHEMBL8308344

Nc1ccc2c(CCC(=O)O)c(C(=O)c3ccc(Cl)cc3)oc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
MAPT P10636 4/20 0.47
KDM4E B2RXH2 4/20 0.47
HPGD P15428 4/20 0.47
NPSR1 Q6W5P4 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HTT P42858 2/20 0.47
ALOX12 P18054 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
POLB P06746 3/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
HSD17B10 Q99714 2/20 0.44
TTR P02766 2/20 0.40
GPR17 Q13304 1/20 0.39
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308345 0.91 ALDH1A1 (0.49) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL4437800 0.87 ALDH1A1 (0.52) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL27445439 0.87 SMN1; SMN2 (0.43) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL8553130 0.86 ALDH1A1 (0.38) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL8307605 0.82 MAPK1 (0.39) ALDH1A1MAPTKDM4EHPGDTDP1
SCHEMBL8307013 0.81 ALDH1A1 (0.45) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL8554638 0.78 ALDH1A1 (0.40) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL27445438 0.78 SMN1; SMN2 (0.46) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL8305127 0.78 MCL1 (0.56) ALDH1A1MAPTKDM4EHPGDNPSR1
SCHEMBL8553140 0.77 MAPT (0.39) ALDH1A1MAPTKDM4EHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685475-B1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1999-01-13 EP disclosed
EP-0685474-B1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1998-09-16 EP disclosed
US-5622989-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
US-5565488-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
EP-0685475-A1 Amino-benzofuryl-and thienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed
EP-0685474-A1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed