SCHEMBL4438009

SCHEMBL4438009

O=C(O)C(Cc1ccc(Cl)c(C(F)(F)F)c1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.56
PPARA Q07869 1/20 0.56
IDO1 P14902 2/20 0.51
KDR P35968 1/20 0.51
FFAR1 O14842 1/20 0.51
PDK1 Q15118 1/20 0.47
ABCB11 O95342 1/20 0.46
FAAH O00519 1/20 0.45
MMP7 P09237 1/20 0.45
CASR P41180 1/20 0.45
KDM4A O75164 1/20 0.44
KDM5A P29375 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
LDHA P00338 1/20 0.44
PYCR1 P32322 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4795847 0.88 PPARG (0.53) PPARGPPARAIDO1KDRPDK1
SCHEMBL2908984 0.88 PPARG (0.53) PPARGPPARAIDO1KDRPDK1
SCHEMBL9901109 0.86 SLC7A5 (0.53) PPARGPPARAIDO1KDRPDK1
SCHEMBL5123818 0.84 KDM4E (0.50) PPARGPPARAIDO1KDRPDK1
SCHEMBL4436198 0.82 EPHX1 (0.46) PPARGPPARAFFAR1LDHAP2RX7
SCHEMBL5241165 0.80 IDO1 (0.48) PPARGPPARAIDO1KDRPDK1
SCHEMBL1039107 0.80 IDO1 (0.48) PPARGPPARAIDO1KDRPDK1
SCHEMBL30302148 0.80 RXRA (0.55) PPARGPPARAIDO1KDRPDK1
SCHEMBL1590516 0.80 RXRA (0.55) PPARGPPARAIDO1KDRPDK1
SCHEMBL2424748 0.80 IDO1 (0.45) PPARGPPARAIDO1KDRPYCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137187-A1 PYRAZOLO [1,5-A]PYRIMIDINES AS INHIBITORS OF STEAROYL-COA DESATURASE Inovacia AB (SE) 2009-12-30 EP disclosed
US-20080255153-A1 New compounds BIOVITRUM AB (PUBL) (SE) 2008-10-16 US disclosed
WO-2008116898-A1 PYRAZOLO [1,5-A]PYRIMIDINES AS INHIBITORS OF STEAROYL-COA DESATURASE BIOVITRUM AB (PUBL) (SE) 2008-10-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080255153-A1 New compounds SCD, SCD5, FADS2 PPARG 203/4885PPARA 278/4885IDO1 307/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.