SCHEMBL4439322

SCHEMBL4439322

CC(=O)C(c1ccc(C(F)(F)F)cc1)c1cc(C(C)C)no1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.41
KCNH2 Q12809 1/20 0.39
MAPK14 Q16539 1/20 0.38
LMNA P02545 2/20 0.37
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
GMNN O75496 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTR1A P08908 1/20 0.37
THRB P10828 1/20 0.37
PIM1 P11309 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAOA P21397 1/20 0.37
SLC6A2 P23975 1/20 0.37
HTR2A P28223 1/20 0.37
AGTR1 P30556 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433211 0.84 LMNA (0.41) MAPK14LMNAAKR1C3AKR1C2SMN1; SMN2
SCHEMBL4441781 0.80 MEN1 (0.41) MAPK14LMNAAKR1C3AKR1C2SMN1; SMN2
SCHEMBL4435069 0.77 CES2 (0.41) MAPK14LMNAAKR1C3AKR1C2SMN1; SMN2
SCHEMBL4432946 0.74 FFAR1 (0.42) MAPK14LMNAAKR1C3AKR1C2SMN1; SMN2
SCHEMBL2304585 0.70 ACP3 (0.56) NPC1RAB9ACES2CES1ALDH1A1
SCHEMBL3729711 0.69 KCNH2 (0.53) MCHR1KCNH2LMNASMN1; SMN2RAB9A
SCHEMBL4431561 0.69 AKR1C3 (0.48) AKR1C3AKR1C2PDE2ACES2CES1
SCHEMBL4438527 0.69 CES2 (0.50) AKR1C3AKR1C2SMN1; SMN2CYP1A2CYP3A4
SCHEMBL4432335 0.69 CES2 (0.41) AKR1C3AKR1C2TP53PDE2ACES2
SCHEMBL4435426 0.69 CNR1 (0.40) LMNAAKR1C3AKR1C2SMN1; SMN2PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed