SCHEMBL4433211

SCHEMBL4433211

CC(=O)C(c1ccc(C(F)(F)F)cc1)c1cc(C)no1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
THRB P10828 2/20 0.41
NPC1 O15118 1/20 0.41
GMNN O75496 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
PIM1 P11309 1/20 0.41
CYP2C9 P11712 1/20 0.41
MAOA P21397 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
AGTR1 P30556 1/20 0.41
CCKBR P32239 1/20 0.41
MC4R P32245 1/20 0.41
CYP2C19 P33261 1/20 0.41
THPO P40225 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4439322 0.84 MCHR1 (0.41) LMNATHRBNPC1GMNNTP53
SCHEMBL4435069 0.80 CES2 (0.41) LMNATHRBNPC1GMNNTP53
SCHEMBL4441781 0.80 MEN1 (0.41) LMNATHRBNPC1GMNNTP53
SCHEMBL4432335 0.74 CES2 (0.41) TP53CES2CES1PDE2AAKR1C3
SCHEMBL4432946 0.73 FFAR1 (0.42) LMNATHRBNPC1GMNNTP53
SCHEMBL4435426 0.73 CNR1 (0.40) LMNASMN1; SMN2CES2CES1PDE2A
SCHEMBL2304585 0.72 ACP3 (0.56) NPC1RAB9ACES2CES1ALDH1A1
SCHEMBL4435804 0.72 HSD11B1 (0.45) SMN1; SMN2CES2CES1PDE2A
SCHEMBL4432365 0.71 AKR1C3 (0.43) CES2CES1PDE2AAKR1C3AKR1C2
SCHEMBL4438527 0.71 CES2 (0.50) CYP1A2CYP3A4CYP2C9SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed