SCHEMBL4442191

SCHEMBL4442191

COc1ccc2c(n1)N(CC(O)C[N+]1(C(C)(C)C)CCC(NC(=O)[O-])CC1)C(=O)CC2

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.32
MTNR1B P49286 5/20 0.32
HTR2C P28335 4/20 0.32
HPGDS O60760 1/20 0.32
RIPK1 Q13546 1/20 0.32
CHRM1 P11229 1/20 0.31
CRHR1 P34998 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3670912 0.77 HPGDS (0.32) MTNR1AMTNR1BHTR2CHPGDS
SCHEMBL3333076 0.77 CHRM1 (0.42) MTNR1AMTNR1BHTR2CRIPK1CHRM1
SCHEMBL3328929 0.77 CHRM1 (0.42) MTNR1AMTNR1BHTR2CRIPK1CHRM1
SCHEMBL22168968 0.75 DRD2 (0.40) CHRM1
SCHEMBL4442971 0.75 DRD2 (0.40) CHRM1
SCHEMBL19470005 0.74 RIPK1 (0.33) MTNR1AMTNR1BHTR2CRIPK1CHRM1
SCHEMBL3327481 0.74 HTR2C (0.34) MTNR1AMTNR1BHTR2CRIPK1
SCHEMBL19470010 0.72 CYP2D6 (0.34) MTNR1AMTNR1BHTR2CCHRM1
SCHEMBL19470009 0.72 CYP2D6 (0.34) MTNR1AMTNR1BHTR2CCHRM1
SCHEMBL17515246 0.69 HPGDS (0.33) MTNR1AMTNR1BHTR2CHPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137196-A1 TRICYCLIC NITROGEN CONTAINING COMPOUNDS AS ANTIBACTERIAL AGENTS Glaxo Group Limited (GB) 2009-12-30 EP disclosed
WO-2008128942-A1 TRICYCLIC NITROGEN CONTAINING COMPOUNDS AS ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2008-10-30 WO disclosed