SCHEMBL4443167

SCHEMBL4443167

COc1ccc2cc(CNS(=O)(=O)c3cccc4c(NC(C)=O)cccc34)ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 3/20 0.55
FABP4 P15090 2/20 0.48
USP30 Q70CQ3 2/20 0.47
ALDH1A1 P00352 5/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
SLC2A1 P11166 1/20 0.46
CYP19A1 P11511 1/20 0.46
CCR8 P51685 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
RECQL P46063 1/20 0.45
EDNRA P25101 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4453211 0.92 NSD2 (0.52) NSD2FABP4ALDH1A1CYP19A1CCR8
SCHEMBL4444987 0.91 NSD2 (0.66) NSD2FABP4USP30ALDH1A1KDM4E
SCHEMBL4454907 0.89 CCR8 (0.51) NSD2FABP4CYP19A1CCR8EDNRA
SCHEMBL4453000 0.88 NSD2 (0.53) NSD2FABP4USP30ALDH1A1CCR8
SCHEMBL4444970 0.86 FABP4 (0.56) NSD2FABP4ALDH1A1CCR8GAA
SCHEMBL4445805 0.84 TP53 (0.47) NSD2FABP4ALDH1A1MEN1KMT2A
SCHEMBL4623757 0.84 FABP4 (0.52) NSD2FABP4ALDH1A1KDM4EKMT2A
SCHEMBL4443216 0.84 CCR8 (0.52) NSD2FABP4USP30ALDH1A1CYP19A1
SCHEMBL4443002 0.83 NSD2 (0.80) NSD2FABP4ALDH1A1SLC2A1CYP19A1
SCHEMBL4443345 0.83 CCR8 (0.48) NSD2FABP4USP30ALDH1A1CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547716-B2 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-06-16 US disclosed
EP-1402890-B1 SULFONAMIDE DERIVATIVES INST MED MOLECULAR DESIGN INC (JP) 2008-01-09 EP disclosed
US-20040234622-A1 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2004-11-25 US disclosed
EP-1402890-A1 SULFONAMIDE DERIVATIVES Institute of Medicinal Molecular Design, Inc. (JP) 2004-03-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040234622-A1 Sulfonamide derivatives PCNA, TOP2A, DDB1 NSD2 122/4885FABP4 1925/4885USP30 4114/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.