SCHEMBL4444970

SCHEMBL4444970

COc1ccc(CNS(=O)(=O)c2cccc3c(NC(C)=O)cccc23)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 2/20 0.56
ALDH1A1 P00352 2/20 0.51
NSD2 O96028 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
LMNA P02545 2/20 0.48
MAPT P10636 1/20 0.48
APP P05067 1/20 0.47
ACHE P22303 1/20 0.47
GAA P10253 1/20 0.47
CCR8 P51685 1/20 0.46
LARS1 Q9P2J5 1/20 0.45
EDNRA P25101 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4623757 0.92 FABP4 (0.52) FABP4ALDH1A1NSD2MAPTGAA
SCHEMBL4444610 0.89 FABP4 (0.51) FABP4ALDH1A1NSD2CCR8EDNRA
SCHEMBL4443167 0.86 NSD2 (0.55) FABP4ALDH1A1NSD2MAPTGAA
SCHEMBL4453211 0.86 NSD2 (0.52) FABP4ALDH1A1NSD2SMN1; SMN2MAPT
SCHEMBL4444987 0.86 NSD2 (0.66) FABP4ALDH1A1NSD2LMNAMAPT
SCHEMBL4453000 0.85 NSD2 (0.53) FABP4ALDH1A1NSD2SMN1; SMN2CCR8
SCHEMBL4443345 0.84 CCR8 (0.48) FABP4ALDH1A1NSD2SMN1; SMN2LMNA
SCHEMBL4454907 0.84 CCR8 (0.51) FABP4NSD2CCR8EDNRA
SCHEMBL4445447 0.83 ALDH1A1 (0.46) FABP4ALDH1A1NSD2SMN1; SMN2CCR8
SCHEMBL4452477 0.83 MEN1 (0.48) FABP4LMNAMAPTGAAEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7547716-B2 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-06-16 US disclosed
EP-1402890-B1 SULFONAMIDE DERIVATIVES INST MED MOLECULAR DESIGN INC (JP) 2008-01-09 EP disclosed
US-20040234622-A1 Sulfonamide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2004-11-25 US disclosed
EP-1402890-A1 SULFONAMIDE DERIVATIVES Institute of Medicinal Molecular Design, Inc. (JP) 2004-03-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040234622-A1 Sulfonamide derivatives PCNA, TOP2A, DDB1 FABP4 1925/4885ALDH1A1 980/4885NSD2 122/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.