SCHEMBL4447221

SCHEMBL4447221

CCOC(=O)COc1c(F)cccc1CCNC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 4/20 0.48
ALDH1A1 P00352 3/20 0.43
KMT2A Q03164 3/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
TAAR1 Q96RJ0 3/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 4/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
NPC1 O15118 1/20 0.39
ABCB1 P08183 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6744989 0.81 NLRP3 (0.59) NLRP3ALDH1A1KMT2AMEN1GAA
SCHEMBL18301079 0.75 NLRP3 (0.52) NLRP3ALDH1A1GAAKDM4ESMN1; SMN2
SCHEMBL16792371 0.73 NLRP3 (0.48) NLRP3ALDH1A1KMT2ALMNAMEN1
SCHEMBL20201867 0.71 CYP4F2 (0.56) NLRP3ALDH1A1KMT2ALMNAGAA
SCHEMBL20562586 0.70 MTNR1A (0.49) ALDH1A1KMT2AMEN1SMN1; SMN2NPC1
SCHEMBL15012550 0.70 NLRP3 (0.50) NLRP3ALDH1A1GAAMAPTKDM4E
SCHEMBL4832334 0.69 SMN1; SMN2 (0.43) NLRP3ALDH1A1KMT2ALMNAMEN1
SCHEMBL2058956 0.69 NLRP3 (0.57) NLRP3ALDH1A1KMT2AMEN1GAA
SCHEMBL18301081 0.69 ALDH1A1 (0.45) NLRP3ALDH1A1GAAL3MBTL1KDM4E
SCHEMBL257483 0.68 USP2 (0.58) NLRP3ALDH1A1KMT2ALMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121598-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2009-11-25 EP disclosed
WO-2008076754-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-06-26 WO disclosed