SCHEMBL4447366

SCHEMBL4447366

CCC(CCOc1cc2c(cc1I)CCC2=O)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
TDP1 Q9NUW8 1/20 0.34
CHRM1 P11229 1/20 0.33
TBXA2R P21731 1/20 0.33
PDE4A P27815 1/20 0.33
ADRA1A P35348 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
HIF1A Q16665 1/20 0.33
PPARA Q07869 5/20 0.33
PPARD Q03181 4/20 0.33
PPARG P37231 4/20 0.33
XDH P47989 1/20 0.31
CA2 P00918 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B1 P14061 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4460094 0.86 BRD4 (0.36) BRD4TDP1CYP1A2CYP2C9PPARA
SCHEMBL4460417 0.81 PPARG (0.39) PPARAPPARDPPARGCA2MAPK1
SCHEMBL4458624 0.79 PPARA (0.44) PPARAPPARDPPARG
SCHEMBL4447367 0.75 BRD4 (0.64) BRD4PDE4ACYP1A2
SCHEMBL4447372 0.74 BRD4 (0.34) BRD4PPARAPPARDPPARGHSD17B1
SCHEMBL7974209 0.74 ABCB1 (0.46) PPARAPPARDPPARG
SCHEMBL21052075 0.72 MAOB (0.54) PPARDPPARG
SCHEMBL17043171 0.71 BRD4 (0.41) BRD4MAPK1HSD17B1
SCHEMBL2304117 0.69 KDM4E (0.44) HSD17B1
SCHEMBL4450025 0.69 TSHR (0.36) PPARAPPARDPPARGCA2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7482484-B2 Carboxylic acids and derivatives for the treatment of and preventing diabetes and dyslipidaemia MERCK PATENT GMBH (DE) 2009-01-27 US disclosed