SCHEMBL4450293

SCHEMBL4450293

CCCCc1c(OC)ccc2cc(C3CCCCCC3)sc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.38
CNR2 P34972 10/20 0.37
CNR1 P21554 5/20 0.37
ALDH1A1 P00352 3/20 0.35
TSHR P16473 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
POLB P06746 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
KDM4E B2RXH2 3/20 0.34
HPGD P15428 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MCOLN3 Q8TDD5 1/20 0.33
MAPT P10636 1/20 0.33
HIF1A Q16665 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4442751 0.84 CNR1 (0.38) CNR2CNR1ALDH1A1MAPK1HPGD
SCHEMBL4452191 0.81 ALDH1A1 (0.39) ALDH1A1TSHRMEN1KMT2ALMNA
SCHEMBL19753110 0.69 CHRNA7 (0.39) HTR2AALDH1A1MEN1KMT2ALMNA
SCHEMBL24089462 0.69 ALOX5 (0.46) ALDH1A1TSHRLMNAMAPK1KDM4E
SCHEMBL10729086 0.68 PDGFRB (0.38) HTR2AALDH1A1TSHRMEN1KMT2A
SCHEMBL4441212 0.67 ACMSD (0.36) ALDH1A1KMT2AKDM4EHPGDNPC1
SCHEMBL3365472 0.67 CNR2 (0.42) CNR2CNR1MEN1KMT2A
SCHEMBL22135589 0.66 PDE10A (0.44) LMNAKDM4EMAPTSMN1; SMN2
SCHEMBL10726933 0.66 PDGFRB (0.38) HTR2AALDH1A1TSHRMEN1KMT2A
SCHEMBL20624818 0.66 PDE4A (0.34) CNR2ALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7476691-B2 Sulfamate benzothiophene derivatives as steroid sulfatase inhibitors LABORATOIRE THERAMEX (MC) 2009-01-13 US disclosed