SCHEMBL4452741

SCHEMBL4452741

CC(Cc1ccccn1)N1C(=O)c2ccccc2C1(Cc1ccc(OC2CCC(F)(F)CC2)nc1)C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 1/20 0.36
SCN9A Q15858 5/20 0.36
KCNH2 Q12809 4/20 0.36
SCN5A Q14524 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC5A7 Q9GZV3 1/20 0.36
IP6K1 Q92551 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ACACB O00763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3954661 0.78 MDM2 (0.42) SCN9AKCNH2SCN5A
SCHEMBL4334649 0.76 SCN9A (0.64) SCN9AKCNH2SCN5A
SCHEMBL4334652 0.66 SCN9A (0.54) SCN9AKCNH2SCN5A
SCHEMBL31591606 0.64 LOX (0.43) LNPEPKCNH2ACACB
SCHEMBL4342306 0.64 LOX (0.43) LNPEPKCNH2ACACB
SCHEMBL3961394 0.62 SCN9A (0.53) SCN9AKCNH2SCN5ACYP3A4
SCHEMBL12367594 0.59 LIPE (0.41)
SCHEMBL5531111 0.59 ALDH1A1 (0.58) KCNH2SLC5A7L3MBTL1
SCHEMBL13568301 0.56 SCN9A (0.58) SCN9AKCNH2SCN5AL3MBTL1
SCHEMBL4461400 0.56 SCN9A (0.60) SCN9AKCNH2SCN5ACYP2D6L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009145720-A1 ISOINDOLINE DERIVATIVES COMPRISING ADDITIONAL HETEROCYCLIC GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO disclosed