SCHEMBL445343

SCHEMBL445343

COC(=O)C(C)(F)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.41
KCNN4 O15554 1/20 0.37
ALDH1A1 P00352 4/20 0.36
TSHR P16473 2/20 0.36
PTPN1 P18031 1/20 0.33
SRC P12931 1/20 0.33
CA2 P00918 1/20 0.32
TP53 P04637 1/20 0.32
CTRB1 P17538 1/20 0.32
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
ELANE P08246 1/20 0.31
CYP2C19 P33261 1/20 0.31
GAA P10253 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9345959 0.86 DGAT1 (0.46) DGAT1KCNN4ALDH1A1TSHRSRC
SCHEMBL28296434 0.79 ALDH1A1 (0.36) ALDH1A1TSHR
SCHEMBL17281569 0.77 DGAT1 (0.39) DGAT1KCNN4ALDH1A1TSHRCA2
SCHEMBL18630822 0.77 DGAT1 (0.44) DGAT1ALDH1A1TSHR
SCHEMBL18630824 0.77 DGAT1 (0.44) DGAT1ALDH1A1TSHR
SCHEMBL4427911 0.76
SCHEMBL21393608 0.76 KCNN4 (0.38) DGAT1KCNN4ALDH1A1TSHRPTPN1
Trifluoroacetic Acid SCHEMBL28075338 0.76 KCNN4 (0.38) DGAT1KCNN4ALDH1A1TSHRPTPN1
SCHEMBL20564537 0.75 DGAT1 (0.38) DGAT1KCNN4ALDH1A1TSHRPTPN1
SCHEMBL135961 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111635312-A Synthesis method of (E) -2-fluoroalkyl-3-butenoate compound 安阳师范学院 2020-09-08 CN claimed
CN-111635312-B Synthesis method of (E) -2-fluoroalkyl-3-butenoate compound 安阳师范学院 2023-02-21 CN disclosed
CN-115461120-A Sulfonylimide compounds as NLRP3 modulators 豪夫迈·罗氏有限公司 2022-12-09 CN disclosed
CN-110627718-B Synthesis method of (E) -beta-monofluoroalkyl-beta, gamma-unsaturated amide 安阳师范学院 2022-10-04 CN disclosed
US-20220227696-A1 Multifunctional Fluorinated Compound, Fluorinated Polymers Made from the Compound, and Related Methods 3M INNOVATIVE PROPERTIES COMPANY 2022-07-21 US disclosed
EP-3980433-A1 MULTIFUNCTIONAL FLUORINATED COMPOUND, FLUORINATED POLYMERS MADE FROM THE COMPOUND, AND RELATED METHODS 3M Innovative Properties Company (US) 2022-04-13 EP disclosed
CN-113906038-A Multifunctional fluorinated compounds, fluorinated polymers made therefrom, and related methods 3M创新有限公司 2022-01-07 CN disclosed
WO-2020245724-A1 MULTIFUNCTIONAL FLUORINATED COMPOUND, FLUORINATED POLYMERS MADE FROM THE COMPOUND, AND RELATED METHODS 3M INNOVATIVE PROPERTIES COMPANY (US) 2020-12-10 WO disclosed
CN-111635312-A Synthesis method of (E) -2-fluoroalkyl-3-butenoate compound 安阳师范学院 2020-09-08 CN disclosed
EP-2481735-A1 Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterials Pfizer Inc. (US) 2012-08-01 EP disclosed
US-20120065188-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC 2012-03-15 US disclosed
US-20110092480-A1 Substituted Heterocyclic Derivatives and Their Pharmaceutical Use and Compositions PFIZER INC. 2011-04-21 US disclosed
EP-2155716-A2 SUBSTITUTED HETEROCYCLIC DERIVATIVES AND COMPOSITIONS AND THEIR PHARMACEUTICAL USE AS ANTIBACTERIALS Pfizer Inc. (US) 2010-02-24 EP disclosed
WO-2008139288-A2 SUBSTITUTED HETEROCYCLIC DERIVATIVES AND COMPOSITIONS AND THEIR PHARMACEUTICAL USE AS ANTIBACTERIALS PFIZER INC. (US) 2008-11-20 WO disclosed
US-20080280879-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC 2008-11-13 US disclosed
EP-0334966-B1 PROCESS FOR SYNTHESIZING OPTICALLY ACTIVE COMPOUNDS NGK INSULATORS LTD (JP) 1994-08-24 EP disclosed
EP-0334966-A1 PROCESS FOR SYNTHESIZING OPTICALLY ACTIVE COMPOUNDS NGK INSULATORS, LTD. (JP) 1989-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120065188-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS XDH, CYP2D6, F12 DGAT1 4831/4885KCNN4 1234/4885ALDH1A1 3777/4885
US-20220227696-A1 Multifunctional Fluorinated Compound, Fluorinated Polymers Made from the Compound, and Related Methods NR1H2, NR1H3, NR1I2 DGAT1 1655/4885KCNN4 855/4885ALDH1A1 2744/4885
US-20080280879-A1 SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS XDH, CYP2D6, F12 DGAT1 4831/4885KCNN4 1234/4885ALDH1A1 3777/4885
US-20110092480-A1 Substituted Heterocyclic Derivatives and Their Pharmaceutical Use and Compositions XDH, CYP2D6, F12 DGAT1 4831/4885KCNN4 1234/4885ALDH1A1 3777/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.