SCHEMBL4454027

SCHEMBL4454027

Nc1c(N)n(-c2ccccc2Cl)c(=S)[nH]c1=O.Nc1c(N=O)c(=O)[nH]c(=S)n1-c1ccccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
KDM4E B2RXH2 4/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
HCAR1 Q9BXC0 4/20 0.38
PDE7A Q13946 1/20 0.36
HPGD P15428 1/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
CASP6 P55212 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ADORA3 P0DMS8 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4498723 0.95 ALDH1A1 (0.44) ALDH1A1KDM4ESMN1; SMN2HCAR1PDE7A
SCHEMBL4498921 0.90 ALDH1A1 (0.48) ALDH1A1KDM4ESMN1; SMN2HCAR1PDE7A
SCHEMBL4465222 0.80 MAPT (0.43) ALDH1A1KDM4ESMN1; SMN2GRIN2DGRIN3B
SCHEMBL4471023 0.80 MEN1 (0.44) ALDH1A1KDM4EHPGDKMT2AMAPT
SCHEMBL4454520 0.77 MAPT (0.47) ALDH1A1KDM4EHPGDKMT2AMAPT
SCHEMBL15330466 0.74 ALDH1A1 (0.44) ALDH1A1KDM4ESMN1; SMN2HCAR1PDE7A
SCHEMBL4492126 0.74 MAPT (0.47) ALDH1A1KDM4ESMN1; SMN2GRIN2DGRIN3B
SCHEMBL4566658 0.74 CA12 (0.38) ALDH1A1KDM4ESMN1; SMN2HPGDKMT2A
SCHEMBL4501815 0.73 MEN1 (0.47) ALDH1A1KDM4EHPGDKMT2AMAPT
SCHEMBL4458183 0.72 GRIN2D (0.38) KDM4EGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010534-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO AstraZeneca AB (SE) 2009-01-07 EP disclosed
WO-2007120097-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO ASTRAZENECA AB (SE) 2007-10-25 WO disclosed