SCHEMBL4456350

SCHEMBL4456350

O=C(O)Nc1cccc(-c2cn[nH]n2)c1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.62
METAP2 P50579 8/20 0.60
IDO1 P14902 9/20 0.56
KEAP1 Q14145 1/20 0.53
SIRT3 Q9NTG7 1/20 0.47
MAPT P10636 1/20 0.47
APOBEC3G Q9HC16 1/20 0.46
ERAP1 Q9NZ08 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22363550 0.78 XDH (1.00) XDH
SCHEMBL21904932 0.75 CYP1A2 (0.57) KMT2A
SCHEMBL28741907 0.75 METAP2 (0.63) XDHMETAP2IDO1KEAP1SIRT3
SCHEMBL29626795 0.75 METAP2 (0.63) XDHMETAP2IDO1KEAP1SIRT3
SCHEMBL13994029 0.75 METAP2 (0.58) XDHMETAP2IDO1KEAP1SIRT3
SCHEMBL28741748 0.75 IDO1 (0.58) XDHMETAP2IDO1KEAP1SIRT3
SCHEMBL21904995 0.74 BTK (0.47) KMT2A
SCHEMBL30331540 0.73 MGLL (0.78)
SCHEMBL7511547 0.73 MGLL (0.78)
SCHEMBL25440056 0.73 MGLL (0.56) MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009090548-A2 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES AS VANILLOID RECEPTOR LIGANDS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-07-23 WO disclosed