SCHEMBL4458062

SCHEMBL4458062

Cn1ccc(-c2cccc([N+](=O)[O-])c2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
MAPT P10636 5/20 0.53
ALDH1A1 P00352 4/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
RAB9A P51151 4/20 0.53
NPC1 O15118 3/20 0.53
PKM P14618 1/20 0.53
IDO1 P14902 1/20 0.52
LMNA P02545 2/20 0.52
KMT2A Q03164 2/20 0.51
KEAP1 Q14145 5/20 0.51
NFE2L2 Q16236 5/20 0.51
GABRA1 P14867 1/20 0.50
GABRB2 P47870 1/20 0.50
THRB P10828 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27774399 0.81 GABRA1 (0.48) CASP3SENP8SENP7SENP6MAPT
SCHEMBL4629018 0.80 KEAP1 (0.55) CASP3SENP7SENP6MAPTALDH1A1
SCHEMBL15392669 0.77 KEAP1 (0.48) CASP3SENP8SENP7SENP6MAPT
SCHEMBL4449942 0.76 ALDH1A1 (0.52) CASP3SENP8SENP7SENP6MAPT
SCHEMBL18985787 0.76 MAPT (0.60) MAPTALDH1A1PKMLMNAKMT2A
SCHEMBL24259133 0.76 KEAP1 (0.53) CASP3SENP8SENP7SENP6MAPT
SCHEMBL4720647 0.76 KEAP1 (0.55) CASP3SENP7MAPTALDH1A1SMN1; SMN2
SCHEMBL6738366 0.75 TSHR (0.76) MAPTALDH1A1SMN1; SMN2RAB9ANPC1
SCHEMBL30461135 0.75 RAB9A (0.69) CASP3SENP8SENP7SENP6MAPT
SCHEMBL30461136 0.75 RAB9A (0.69) CASP3SENP8SENP7SENP6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022228547-A1 PHOSPHONYL DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL APPLICATION THEREOF 四川海思科制药有限公司 2022-11-03 WO disclosed
WO-2009090548-A2 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES AS VANILLOID RECEPTOR LIGANDS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-07-23 WO disclosed