SCHEMBL4460265

SCHEMBL4460265

O=C(Nc1cccc2c1C(=O)NC2=O)NC1C2CN(c3ccc(F)cc3F)CC21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.44
KDM4E B2RXH2 8/20 0.44
HPGD P15428 3/20 0.44
HSD17B10 Q99714 3/20 0.44
GAA P10253 3/20 0.44
CASP3 P42574 4/20 0.43
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
MAPK10 P53779 1/20 0.41
POLB P06746 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TRPV1 Q8NER1 3/20 0.38
MAPT P10636 1/20 0.38
CASP1 P29466 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13783924 1.00 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL4460262 1.00 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL4472460 0.86 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL13783798 0.86 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL4472454 0.86 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL4451601 0.81 CASP3 (0.43) ALDH1A1KDM4EHPGDHSD17B10CASP3
SCHEMBL13783979 0.81 CASP3 (0.43) ALDH1A1KDM4EHPGDHSD17B10CASP3
SCHEMBL4451608 0.81 CASP3 (0.43) ALDH1A1KDM4EHPGDHSD17B10CASP3
SCHEMBL4774278 0.79 POLB (0.38) ALDH1A1GAAPOLBMEN1KMT2A
SCHEMBL4455115 0.77 ALDH1A1 (0.40) ALDH1A1KDM4EHSD17B10GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009090548-A2 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES AS VANILLOID RECEPTOR LIGANDS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-07-23 WO disclosed