SCHEMBL4461012

SCHEMBL4461012

Nc1ccccc1-n1nccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.48
KDM4E B2RXH2 3/20 0.48
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
USP2 O75604 2/20 0.45
TP53 P04637 1/20 0.45
HTT P42858 1/20 0.45
KEAP1 Q14145 1/20 0.43
ALDH1A1 P00352 3/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP3A4 P08684 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
ADRA2C P18825 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.36
ATAD2 Q6PL18 1/20 0.35
POLB P06746 1/20 0.34
TSHR P16473 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10622430 0.74 KDM4E (0.48) GAAKDM4EMEN1KMT2AUSP2
SCHEMBL19480734 0.73 NOS3 (0.45) GAAKDM4EMEN1KMT2AUSP2
SCHEMBL19480727 0.73 MAPT (0.42) GAAKDM4EMEN1KMT2AHTT
SCHEMBL26386600 0.71 MGLL (0.43) NPC1CYP19A1
SCHEMBL2829025 0.71 IDO1 (0.48) GAAKDM4EMEN1KMT2AHTT
SCHEMBL17145963 0.71 MGLL (0.43) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL7729323 0.71 GAA (0.39) GAAKDM4EMEN1KMT2AUSP2
SCHEMBL1531523 0.71 MAPK1 (0.56) GAAKDM4EMEN1KMT2AUSP2
SCHEMBL20551340 0.70 SMN1; SMN2 (0.46) GAAKDM4EMEN1KMT2ATP53
SCHEMBL20766782 0.70 HCRTR1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014060112-A1 PYRAZOLO[4,3-D]PYRIMIDINES AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2014-04-24 WO disclosed
WO-2009090548-A2 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES AS VANILLOID RECEPTOR LIGANDS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-07-23 WO disclosed