SCHEMBL4462380

SCHEMBL4462380

COc1c(C(C)(C)C)cc(C(=O)N2CCC(C(N)=O)C2)cc1C(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KCNH2 Q12809 4/20 0.47
PKM P14618 1/20 0.44
PDK2 Q15119 1/20 0.43
HSD17B10 Q99714 2/20 0.43
GAA P10253 2/20 0.43
GLA P06280 1/20 0.43
HPGD P15428 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5633304 0.86 ALDH1A1 (0.53) ALDH1A1KCNH2PKMPDK2HSD17B10
SCHEMBL5633990 0.84 GAA (0.62) ALDH1A1PKMHSD17B10GAAHPGD
SCHEMBL5634807 0.83 ALDH1A1 (0.44) ALDH1A1KCNH2PDK2HSD17B10GAA
SCHEMBL5634575 0.82 KCNH2 (0.54) KCNH2GAAHSP90AA1HSP90AB1
SCHEMBL5397724 0.81 ALDH1A1 (0.56) ALDH1A1PDK2HSD17B10GAAGLA
SCHEMBL4462385 0.81 KCNH2 (0.49) KCNH2PDK2GAAHSP90AA1HSP90AB1
SCHEMBL4599280 0.78 KCNH2 (0.47) ALDH1A1KCNH2PDK2GAAHSP90AA1
SCHEMBL30150598 0.76 POLB (0.68) ALDH1A1HSD17B10GAAGLAHPGD
SCHEMBL5399828 0.76 GAA (0.63) ALDH1A1PDK2HSD17B10GAAGLA
SCHEMBL8605250 0.74 PKM (0.61) ALDH1A1KCNH2PKMGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7507760-B2 N-type calcium channel blockers NEUROMED PHARMACEUTICALS LTD. (CA) 2009-03-24 US claimed
US-7244758-B2 N-type calcium channel blockers NEUROMED PHARMACEUTICALS LTD. (CA) 2007-07-17 US claimed
US-20050014748-A1 N-type calcium channel blockers NEUROMED TECHNOLOGIES INC. 2005-01-20 US claimed
EP-1718633-A1 N-TYPE CALCIUM CHANNEL BLOCKERS Neuromed Pharmaceuticals, Ltd. (CA) 2006-11-08 EP disclosed
WO-2005070919-A1 N-TYPE CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2005-08-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014748-A1 N-type calcium channel blockers CACNA1B, CACNA1C, CACNA1I ALDH1A1 2914/4885KCNH2 33/4885PKM 2560/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.